SCHEMBL6633964

SCHEMBL6633964

Cc1ccc(Sc2ccccc2C(N)=O)s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 2/20 0.54
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
UBE2I P63279 1/20 0.46
SAE1 Q9UBE0 1/20 0.46
UBA2 Q9UBT2 1/20 0.46
MAPT P10636 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
METAP2 P50579 1/20 0.36
ICAM1 P05362 2/20 0.35
SELE P16581 2/20 0.35
PRNP P04156 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NTRK1 P04629 1/20 0.35
BCAT2 O15382 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701766 0.81 SIRT1 (0.54) SIRT1ALDH1A1KDM4EHPGDLMNA
SCHEMBL7707377 0.81 SIRT1 (0.50) SIRT1ALDH1A1KDM4EHPGDLMNA
SCHEMBL3077375 0.77 SIRT1 (0.77) SIRT1ALDH1A1KDM4EHPGDMAPT
SCHEMBL6629448 0.74 SIRT1 (0.57) SIRT1ALDH1A1KDM4EHPGDLMNA
SCHEMBL701691 0.74 SIRT1 (0.60) SIRT1ALDH1A1KDM4EHPGDLMNA
SCHEMBL6632850 0.73 SIRT1 (0.65) SIRT1ALDH1A1KDM4EHPGDLMNA
Iodide SCHEMBL7710889 0.72 SIRT1 (0.58) SIRT1ALDH1A1KDM4EHPGDLMNA
SCHEMBL6633843 0.71 SIRT1 (0.53) SIRT1ALDH1A1KDM4EHPGDMAPT
SCHEMBL1030659 0.71 SIRT1 (1.00) SIRT1ALDH1A1KDM4EHPGDLMNA
SCHEMBL29530768 0.69 SIRT1 (0.64) SIRT1ALDH1A1KDM4EHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480977-A2 SUBSTITUTED ARYL COMPOUNDS FOR TREATMENT OF DISEASE PHARMACIA & UPJOHN COMPANY (US) 2004-12-01 EP claimed
WO-2003070728-A2 AZABICYCLO-SUBSTITUTED BENZOYLAMIDES AND THIOAMIDES FOR TREATMENT OF CNS-RELATED DISORDERS PHARMACIA & UPJOHN COMPANY (US) 2003-08-28 WO claimed
WO-2002016357-A2 QUINUCLIDINE-SUBSTITUTED ARYL MOIETIES FOR TREATMENT OF DISEASE (NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS) PHARMACIA & UPJOHN COMPANY (US) 2002-02-28 WO claimed