SCHEMBL6629665

SCHEMBL6629665

NC(=O)c1cc(-c2ccsc2)ccc1N1CCNCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACMSD Q8TDX5 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
ALOX15 P16050 1/20 0.44
GFER P55789 1/20 0.44
YWHAG P61981 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CHEK1 O14757 2/20 0.43
HTT P42858 1/20 0.43
CDC7 O00311 1/20 0.41
CDK9 P50750 1/20 0.41
MTOR P42345 1/20 0.41
CHEK2 O96017 2/20 0.40
PDPK1 O15530 1/20 0.39
RPS6KB1 P23443 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6631182 0.78 HDAC2 (0.48) KDM4EMEN1MAPTTHRBALOX15
SCHEMBL11217216 0.76 HSD17B10 (0.53) KDM4EMEN1MAPTTHRBALOX15
SCHEMBL4916238 0.75 HTR7 (0.44) MAPTCHEK1MTORALDH1A1SMN1; SMN2
SCHEMBL22542062 0.74 KDM4E (0.51) KDM4EMEN1MAPTTHRBALOX15
SCHEMBL3568654 0.72 KCNH2 (0.61) ACMSDKDM4EMAPTGFERKMT2A
SCHEMBL6605568 0.72 HTR7 (0.51) CHEK1HTR6
SCHEMBL20883677 0.71 KDM4E (0.48) KDM4EMEN1MAPTTHRBALOX15
SCHEMBL6627618 0.71 ADRB2 (0.49) KDM4EMEN1MAPTTHRBALOX15
SCHEMBL3468316 0.71 ACMSD (0.54) ACMSDMAPTCHEK1CHEK2ALDH1A1
SCHEMBL3898554 0.71 ACMSD (0.45) ACMSDMEN1MAPTKMT2ACHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389194-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-02-18 EP disclosed
WO-2002088101-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2002-11-07 WO disclosed