SCHEMBL6632644

SCHEMBL6632644

CN(C#N)C(=O)C(CC1CCCCC1)OC(=O)N1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.47
CTSL P07711 8/20 0.45
CTSB P07858 6/20 0.45
CTSH P09668 3/20 0.45
CTSK P43235 6/20 0.43
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP8 P22894 1/20 0.39
MMP13 P45452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6062499 1.00 CTSS (0.47) CTSSCTSLCTSBCTSHCTSK
SCHEMBL6696441 0.91 CTSK (0.46) CTSSCTSLCTSBCTSHCTSK
SCHEMBL6653241 0.91 CTSK (0.46) CTSSCTSLCTSBCTSHCTSK
SCHEMBL6694050 0.91 CTSK (0.49) CTSSCTSLCTSBCTSHCTSK
SCHEMBL6063838 0.89 CTSS (0.44) CTSSCTSLCTSBCTSHCTSK
SCHEMBL6062906 0.85 HSD11B1 (0.43) CTSSCTSLCTSBCTSHCTSK
SCHEMBL14110478 0.83 CTSS (0.47) CTSSCTSLCTSBCTSHCTSK
SCHEMBL5523879 0.81 CTSS (0.66) CTSSCTSLCTSBCTSHCTSK
SCHEMBL6062496 0.81 CTSS (0.52) CTSSCTSLCTSBCTSK
SCHEMBL6062505 0.81 CTSS (0.52) CTSSCTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397340-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-03-17 EP disclosed
WO-2002098850-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-12-12 WO disclosed