SCHEMBL6632931

SCHEMBL6632931

NC(=O)C1(c2ccccc2)CCNCC1.c1ccc(C2CCNCC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.56
SLC18A3 Q16572 1/20 0.56
OPRM1 P35372 2/20 0.47
OPRL1 P41146 1/20 0.43
HSD11B1 P28845 5/20 0.43
HDAC1 Q13547 1/20 0.41
TACR1 P25103 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
NAMPT P43490 1/20 0.40
JAK3 P52333 1/20 0.40
HTR6 P50406 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL476403 0.87 OPRM1 (0.58) OPRM1OPRL1HSD11B1HDAC1TACR1
Hydrochloric Acid SCHEMBL1990667 0.85 OPRM1 (0.56) OPRM1OPRL1HSD11B1HDAC1TACR1
Trifluoroacetic Acid SCHEMBL16413809 0.78 OPRM1 (0.50) OPRM1OPRL1HSD11B1HDAC1TACR1
SCHEMBL9400647 0.75 SLC18A3 (0.77) SIGMAR1SLC18A3NAMPTJAK3HTR6
SCHEMBL2722547 0.75 AKR1C1 (0.57) OPRM1OPRL1HSD11B1HDAC1
SCHEMBL501923 0.75 AKR1C1 (0.57) OPRM1OPRL1HSD11B1HDAC1
Benzene SCHEMBL28128069 0.74 SLC18A3 (1.00) SIGMAR1SLC18A3HTR6
SCHEMBL4574 0.74 SLC18A3 (1.00) SIGMAR1SLC18A3HTR6
Butanedione SCHEMBL16136715 0.74 SLC18A3 (0.74) SIGMAR1SLC18A3NAMPTJAK3HTR6
SCHEMBL373567 0.73 AKR1C1 (0.68) OPRM1HSD11B1HDAC1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1456200-A1 LACTAMS AS TACHYKININ ANTAGONISTS Pfizer Limited (GB) 2004-09-15 EP disclosed
WO-2003051868-A1 LACTAMS AS TACHYKININ ANTAGONISTS PFIZER LIMITED (GB) 2003-06-26 WO disclosed