SCHEMBL6637293

SCHEMBL6637293

Cc1nn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1-c1ccc2ncc(-c3ccc(S(=O)(=O)N4CCCC4)cc3)n2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
GAA P10253 5/20 0.41
KCNH2 Q12809 1/20 0.41
KDM4E B2RXH2 2/20 0.39
PKM P14618 2/20 0.38
PIK3CA P42336 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 4/20 0.36
LMNA P02545 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPSR1 Q6W5P4 3/20 0.36
HTT P42858 2/20 0.36
KIT P10721 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
FLT3 P36888 1/20 0.35
POLB P06746 2/20 0.35
TNF P01375 1/20 0.35
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3846968 0.86 KCNH2 (0.44) KCNH2PIK3CATSHRLMNAFLT3
SCHEMBL3846693 0.79 PGR (0.39) ALDH1A1KCNH2KDM4EPIK3CAMEN1
SCHEMBL3849695 0.77 TGFBR1 (0.37) KCNH2PIK3CAMEN1KMT2ALMNA
SCHEMBL3850040 0.76 FLT3 (0.45) KCNH2FLT3TGFBR1
Hydrochloric Acid SCHEMBL3847228 0.76 ALDH1A1 (0.42) ALDH1A1GAAKCNH2KDM4EPKM
SCHEMBL3852869 0.75 TGFBR1 (0.38) TGFBR1
SCHEMBL3845703 0.74 TGFBR1 (0.41) KCNH2TGFBR1
SCHEMBL3846455 0.74 FLT3 (0.51) KCNH2FLT3TGFBR1
SCHEMBL3849014 0.73 AKT1 (0.41) KCNH2PIK3CAFLT3TGFBR1
SCHEMBL3848269 0.72 KCNH2 (0.48) KCNH2PIK3CAKITFLT3TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed