SCHEMBL6637355

SCHEMBL6637355

CCCCCOc1ccccc1C1C(C#N)=C(C)NC(=O)N1C(=O)NCC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 6/20 0.42
TSHR P16473 4/20 0.41
ALDH1A1 P00352 11/20 0.41
GAA P10253 6/20 0.41
MAPT P10636 4/20 0.41
MAPK1 P28482 2/20 0.41
MEN1 O00255 2/20 0.41
TP53 P04637 3/20 0.40
THRB P10828 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
HIF1A Q16665 2/20 0.38
POLB P06746 2/20 0.38
NPSR1 Q6W5P4 4/20 0.38
HSD17B10 Q99714 3/20 0.38
KDM4E B2RXH2 3/20 0.38
GLA P06280 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6640675 0.89 LMNA (0.48) KMT2AHTTLMNATSHRALDH1A1
SCHEMBL6321486 0.79 CACNA1F (0.46)
SCHEMBL6320957 0.74 ADRA1D (0.41) LMNAMAPTCYP3A4CYP2C9CYP2C19
SCHEMBL6312439 0.74 ALDH1A1 (0.45) KMT2ALMNATSHRALDH1A1GAA
SCHEMBL6314298 0.72 HPGD (0.43) HTTLMNAALDH1A1GAAMAPT
SCHEMBL6313974 0.71 CACNA1C (0.35) KMT2AHTTLMNATSHRALDH1A1
SCHEMBL6318791 0.70 ELANE (0.46) TSHRALDH1A1ALOX15
SCHEMBL6314301 0.70 ABCC9 (0.45)
SCHEMBL6321556 0.70 CACNA1C (0.41) KMT2AHTTLMNATSHRALDH1A1
SCHEMBL6137193 0.63 CACNA1F (0.43) KMT2ALMNATSHRALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373223-A4 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL MYERS SQUIBB CO (US) 2004-09-29 EP disclosed
EP-1373223-A1 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES Bristol-Myers Squibb Company (US) 2004-01-02 EP disclosed
WO-2002079169-A1 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-10-10 WO disclosed