SCHEMBL6645425

SCHEMBL6645425

N#Cc1ccc2c(c1)C1CCCC1C(N)=N2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 20/20 1.00
NOS2 P35228 18/20 1.00
NOS3 P29474 17/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6646269 0.88 NOS1 (0.79) NOS1NOS2NOS3
SCHEMBL6642217 0.77 NOS1 (1.00) NOS1NOS2NOS3
SCHEMBL6644308 0.77 NOS1 (1.00) NOS1NOS2NOS3
SCHEMBL6644598 0.73 NOS1 (1.00) NOS1NOS2NOS3
SCHEMBL6646137 0.72 NOS3 (0.56) NOS1NOS2NOS3
SCHEMBL6646955 0.71 NOS1 (1.00) NOS1NOS2NOS3
SCHEMBL6639670 0.70 NOS1 (0.60) NOS1NOS2NOS3
SCHEMBL6643315 0.69 NOS1 (1.00) NOS1NOS2NOS3
SCHEMBL6137675 0.68 NOS3 (0.67) NOS1NOS2NOS3
SCHEMBL6643807 0.68 NOS1 (1.00) NOS1NOS2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6391887-B1 ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASE; CARDIOVASCULAR DISORDERS SCHERING AKTIENGESELLSCHAFT (DE) 2002-05-21 US claimed
EP-1054869-B1 3,4-DIHYDROQUINOLINE DERIVATIVES AS NITROGEN MONOXIDE SYNTHASE (NOS) INHIBITORS SCHERING AG (DE) 2004-09-22 EP disclosed
US-6391887-B1 ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASE; CARDIOVASCULAR DISORDERS SCHERING AKTIENGESELLSCHAFT (DE) 2002-05-21 US disclosed