SCHEMBL6648546

SCHEMBL6648546

CCc1ccncc1-c1nc(-c2cccc([N+](=O)[O-])c2)cs1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOA P21397 10/20 0.52
MAOB P27338 10/20 0.52
MAPT P10636 4/20 0.49
ALDH1A1 P00352 4/20 0.49
LMNA P02545 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
EIF4E P06730 1/20 0.48
CSNK2A1 P68400 1/20 0.48
RAB9A P51151 3/20 0.48
NPC1 O15118 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GAA P10253 1/20 0.47
VCP P55072 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6646934 0.94 MAOA (0.50) MAOAMAOBMAPTALDH1A1LMNA
SCHEMBL6646928 0.84 MAPT (0.48) MAOAMAOBMAPTALDH1A1LMNA
SCHEMBL6646768 0.82 CYP19A1 (0.56) MAPTALDH1A1MEN1KMT2AEIF4E
SCHEMBL6804280 0.82 CYP19A1 (0.68) MAPTALDH1A1RAB9ANPC1GAA
SCHEMBL6652389 0.81 KDM4E (0.59) ALDH1A1KMT2ARAB9ANPC1
SCHEMBL6649196 0.81 C1S (0.55) MAPTALDH1A1LMNAMEN1KMT2A
SCHEMBL6653028 0.81 MAPT (0.50) MAOAMAOBMAPTALDH1A1LMNA
Bromide SCHEMBL7079674 0.81 CYP19A1 (0.66) MAPTALDH1A1MEN1KMT2ARAB9A
SCHEMBL6649515 0.79 MAPT (0.51) MAOAMAOBMAPTALDH1A1LMNA
SCHEMBL6651011 0.79 EIF4E (0.48) MAPTEIF4ERAB9ANPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432706-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
WO-2003027085-A2 3-PYRIDYL OR 4-ISOQUINOLINYL THIAZOLES AS C17,20 LYASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed