SCHEMBL6649239

SCHEMBL6649239

CN(C)CCCOc1cc(Cl)ccc1Cc1nccn1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM5 Q9NZQ8 1/20 0.49
HRH1 P35367 1/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.38
NR4A2 P43354 2/20 0.37
HPGD P15428 2/20 0.37
MAPK1 P28482 2/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
CYP2C19 P33261 1/20 0.37
THPO P40225 1/20 0.37
RAB9A P51151 1/20 0.37
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675930 0.94 TRPM5 (0.50) TRPM5KMT2AKDM4ENR4A2MAPK1
SCHEMBL6654159 0.85 TRPM5 (0.40) TRPM5HRH1KMT2AKDM4EMAPK1
SCHEMBL6648694 0.82 TRPM5 (0.38) TRPM5HRH1KMT2AKDM4EMAPK1
SCHEMBL6651875 0.81 SMN1; SMN2 (0.48) TRPM5HRH1KDM4ENPC1RAB9A
SCHEMBL6650448 0.80 TRPM5 (0.41) TRPM5KMT2AKDM4ENR4A2MAPK1
SCHEMBL6653862 0.79 CYP1A2 (0.35) TRPM5HRH1KMT2AKDM4EALDH1A1
SCHEMBL6654254 0.78 TRPM5 (0.37) TRPM5KMT2AKDM4ENR4A2HPGD
SCHEMBL6650011 0.76 DRD4 (0.40) HRH1KDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL6650126 0.75 DRD4 (0.34) TRPM5HRH1KMT2ACYP1A2CYP3A4
SCHEMBL6654434 0.74 DRD4 (0.37) TRPM5HRH1KMT2AKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103243-B1 UTILIZATION OF ARYL(OR HETEROARYL)AZOLYLCARBINOL DERIVATIVES FOR THE TREATMENT OF TROUBLES MEDIATED BY AN EXCESS OF SUBSTANCE P ESTEVE LABOR DR (ES) 2004-01-07 EP claimed