SCHEMBL6654434

SCHEMBL6654434

CN(C)CCCOCc1cccc(Cc2nccn2C)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.37
HRH1 P35367 2/20 0.36
SLC6A4 P31645 2/20 0.35
HRH3 Q9Y5N1 2/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
KDM4E B2RXH2 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1B P28222 1/20 0.33
TRPM5 Q9NZQ8 1/20 0.32
GUCY1B2 O75343 1/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651100 0.87 HRH3 (0.38) DRD4HRH1SLC6A4HRH3CYP1A2
SCHEMBL6654159 0.83 TRPM5 (0.40) DRD4HRH1SLC6A4HRH3CYP1A2
SCHEMBL6650126 0.82 DRD4 (0.34) DRD4HRH1HRH3CYP1A2CYP2D6
SCHEMBL6650011 0.81 DRD4 (0.40) DRD4HRH1HRH3CYP1A2CYP2D6
SCHEMBL6649431 0.80 DRD4 (0.37) DRD4HRH3LMNAMEN1KMT2A
SCHEMBL6653862 0.77 CYP1A2 (0.35) DRD4HRH1HRH3CYP1A2CYP2D6
SCHEMBL6650448 0.76 TRPM5 (0.41) KDM4ELMNAMEN1KMT2ATRPM5
SCHEMBL6672746 0.75 DRD4 (0.39) DRD4CYP1A2CYP2D6KDM4ECYP2C9
SCHEMBL6672324 0.75 KDM4E (0.33) DRD4CYP1A2CYP2D6KDM4ECYP2C9
SCHEMBL6649239 0.74 TRPM5 (0.49) HRH1CYP1A2CYP2D6KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103243-B1 UTILIZATION OF ARYL(OR HETEROARYL)AZOLYLCARBINOL DERIVATIVES FOR THE TREATMENT OF TROUBLES MEDIATED BY AN EXCESS OF SUBSTANCE P ESTEVE LABOR DR (ES) 2004-01-07 EP claimed