SCHEMBL6651100

SCHEMBL6651100

CN(C)CCCOCc1c(Cl)cccc1Cc1nccn1C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.38
DRD4 P21917 1/20 0.38
HRH1 P35367 1/20 0.35
MC4R P32245 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
SLC6A4 P31645 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
HSD11B1 P28845 1/20 0.32
LMNA P02545 1/20 0.32
ALK Q9UM73 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
FGFR1 P11362 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6649431 0.93 DRD4 (0.37) HRH3DRD4MC4RTAAR1LMNA
SCHEMBL6650126 0.87 DRD4 (0.34) HRH3DRD4HRH1CYP1A2CYP3A4
SCHEMBL6654434 0.87 DRD4 (0.37) HRH3DRD4HRH1CYP1A2CYP3A4
SCHEMBL6650011 0.84 DRD4 (0.40) HRH3DRD4HRH1CYP1A2CYP3A4
SCHEMBL6672324 0.80 KDM4E (0.33) DRD4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6654159 0.79 TRPM5 (0.40) HRH3DRD4HRH1MC4RCYP1A2
SCHEMBL6672746 0.78 DRD4 (0.39) DRD4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6653862 0.75 CYP1A2 (0.35) HRH3DRD4HRH1CYP1A2CYP3A4
SCHEMBL6648324 0.75 MC4R (0.41) DRD4MC4RTAAR1MEN1KMT2A
SCHEMBL6649239 0.73 TRPM5 (0.49) HRH1CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103243-B1 UTILIZATION OF ARYL(OR HETEROARYL)AZOLYLCARBINOL DERIVATIVES FOR THE TREATMENT OF TROUBLES MEDIATED BY AN EXCESS OF SUBSTANCE P ESTEVE LABOR DR (ES) 2004-01-07 EP claimed