SCHEMBL6651171

SCHEMBL6651171

Nc1cc(-c2cccc(C(F)(F)F)c2)ccc1N1CCNCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
HTR2C P28335 3/20 0.56
HTR3A P46098 2/20 0.56
HTR3E A5X5Y0 1/20 0.56
HTR3B O95264 1/20 0.56
HTR1D P28221 1/20 0.56
HTR3D Q70Z44 1/20 0.56
HTR3C Q8WXA8 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
MAPT P10636 2/20 0.55
THRB P10828 1/20 0.55
KDM4E B2RXH2 1/20 0.50
LMNA P02545 1/20 0.50
IDH2 P48735 1/20 0.47
ASIC3 Q9UHC3 1/20 0.47
ADRB2 P07550 1/20 0.44
NCF1 P14598 1/20 0.44
HTR1A P08908 3/20 0.44
ADRB1 P08588 2/20 0.44
HTR7 P34969 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6627622 0.84 ALDH1A1 (0.68) ALDH1A1HTR2CHTR3AHTR3EHTR3B
SCHEMBL14341303 0.81 HTR2C (0.70) ALDH1A1HTR2CHTR3AHTR3EHTR3B
SCHEMBL6630046 0.80 ALDH1A1 (0.61) ALDH1A1HTR2CHTR3AHTR3EHTR3B
SCHEMBL5566823 0.78 HTR7 (0.63) ALDH1A1HTR2CHTR3AHTR3EHTR3B
SCHEMBL9401046 0.75 ALDH1A1 (0.57) ALDH1A1HTR2CHTR3AHTR3EHTR3B
SCHEMBL6712209 0.74 HTR2C (0.55) ALDH1A1HTR2CHTR3AHTR3EHTR3B
SCHEMBL6631185 0.74 CYP1A2 (0.52) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL4907297 0.74 HTR2C (0.63) ALDH1A1HTR2CHTR3AHTR3EHTR3B
SCHEMBL6629232 0.73 ADRB1 (0.53) ALDH1A1HTR3AHTR3EHTR3BHTR3D
SCHEMBL28338201 0.73 ALDH1A1 (0.78) ALDH1A1MAPTKDM4ELMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389194-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-02-18 EP disclosed
WO-2002088101-A2 INHIBITORS OF BACE VERTEX PHARMACEUTICALS INCORPORATED (US) 2002-11-07 WO disclosed