SCHEMBL6652771

SCHEMBL6652771

COc1ccnc(N2CCN(C(=O)c3ccncc3)CC2)n1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
GAA P10253 1/20 0.57
SLC6A7 Q99884 6/20 0.56
PARP1 P09874 1/20 0.54
KDM4E B2RXH2 2/20 0.53
HPGD P15428 1/20 0.53
TSHR P16473 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
GBA1 P04062 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
HCRTR1 O43613 1/20 0.49
HCRTR2 O43614 1/20 0.49
DRD3 P35462 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PKM P14618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6653359 0.99 ALDH1A1 (0.56) ALDH1A1GAASLC6A7PARP1KDM4E
SCHEMBL6653362 0.96 ALDH1A1 (0.54) ALDH1A1GAASLC6A7PARP1KDM4E
SCHEMBL6655484 0.91 SLC6A7 (0.62) ALDH1A1SLC6A7PARP1KDM4EHPGD
SCHEMBL6652211 0.89 SLC6A7 (0.62) ALDH1A1SLC6A7PARP1KDM4EHPGD
SCHEMBL6652154 0.89 L3MBTL1 (0.67) ALDH1A1SLC6A7PARP1KDM4EHPGD
SCHEMBL6651715 0.88 SLC6A7 (0.65) ALDH1A1GAASLC6A7PARP1KDM4E
Hydrochloric Acid SCHEMBL6653082 0.88 SLC6A7 (0.61) ALDH1A1SLC6A7PARP1KDM4EHPGD
Hypochlorous Acid SCHEMBL6653089 0.88 SLC6A7 (0.61) ALDH1A1SLC6A7PARP1KDM4EHPGD
Hydrochloric Acid SCHEMBL6650956 0.88 L3MBTL1 (0.65) ALDH1A1SLC6A7PARP1KDM4EHPGD
Hydrochloric Acid SCHEMBL6657431 0.87 SLC6A7 (0.64) ALDH1A1GAASLC6A7PARP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006110-B1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-02-11 EP claimed
US-6372746-B1 ANTICONVULSIVE AGENTS, SEDATIVES AND EATING DISORDERS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2002-04-16 US claimed
EP-1006110-A1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2000-06-07 EP claimed