SCHEMBL6655484

SCHEMBL6655484

COc1ccnc(N2CCN(C(=O)c3ccccc3)CC2)n1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 10/20 0.62
PKM P14618 1/20 0.58
ALDH1A1 P00352 2/20 0.58
HPGD P15428 1/20 0.58
TSHR P16473 1/20 0.57
PARP1 P09874 1/20 0.55
KDM4E B2RXH2 2/20 0.55
HCRTR1 O43613 2/20 0.54
HCRTR2 O43614 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6652771 0.91 ALDH1A1 (0.57) SLC6A7PKMALDH1A1HPGDTSHR
Hydrochloric Acid SCHEMBL6653359 0.90 ALDH1A1 (0.56) SLC6A7PKMALDH1A1HPGDTSHR
SCHEMBL6651764 0.88 ALDH1A1 (0.59) SLC6A7ALDH1A1HPGDPARP1KDM4E
SCHEMBL6653362 0.88 ALDH1A1 (0.54) SLC6A7ALDH1A1HPGDTSHRPARP1
SCHEMBL6652154 0.88 L3MBTL1 (0.67) SLC6A7ALDH1A1HPGDPARP1KDM4E
SCHEMBL6652211 0.88 SLC6A7 (0.62) SLC6A7ALDH1A1HPGDPARP1KDM4E
Hydrochloric Acid SCHEMBL6656739 0.87 ALDH1A1 (0.58) SLC6A7ALDH1A1HPGDPARP1KDM4E
SCHEMBL6653885 0.87 ALDH1A1 (0.79) SLC6A7ALDH1A1HPGDKDM4EL3MBTL1
Hydrochloric Acid SCHEMBL6653082 0.87 SLC6A7 (0.61) SLC6A7ALDH1A1HPGDPARP1KDM4E
SCHEMBL6657811 0.87 HCRTR1 (0.59) SLC6A7ALDH1A1PARP1KDM4EHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1202087-C Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments ESTEVE LABOR DR (ES) 2005-05-18 CN claimed
EP-1006110-B1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-02-11 EP claimed
US-6372746-B1 ANTICONVULSIVE AGENTS, SEDATIVES AND EATING DISORDERS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2002-04-16 US claimed
CN-1268124-A Acyl-piperazinyl-pyrimidine derivatives, their preparation and use as medicaments ESTEVE LABOR DR (ES) 2000-09-27 CN claimed
EP-1006110-A1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2000-06-07 EP claimed
CN-1202087-C Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments ESTEVE LABOR DR (ES) 2005-05-18 CN disclosed
EP-1006110-B1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-02-11 EP disclosed
US-6372746-B1 ANTICONVULSIVE AGENTS, SEDATIVES AND EATING DISORDERS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2002-04-16 US disclosed
CN-1268124-A Acyl-piperazinyl-pyrimidine derivatives, their preparation and use as medicaments ESTEVE LABOR DR (ES) 2000-09-27 CN disclosed
EP-1006110-A1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2000-06-07 EP disclosed