SCHEMBL6658083

SCHEMBL6658083

CC[C@@]1(C(=O)N2CCN(Cc3ccc(OC)cc3)CC2)CCCCN1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
PKM P14618 1/20 0.50
ALDH1A1 P00352 1/20 0.47
FAAH O00519 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.45
LSS P48449 1/20 0.45
SIGMAR1 Q99720 2/20 0.45
TSHR P16473 2/20 0.45
USP2 O75604 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
CYP2D6 P10635 1/20 0.43
PARP1 P09874 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6659277 0.84 HSD11B1 (0.50) POLBALDH1A1SMN1; SMN2TSHRCYP1A2
Hydrochloric Acid SCHEMBL6659375 0.76 SMN1; SMN2 (0.53) PKMALDH1A1SMN1; SMN2SIGMAR1HTT
Hydrochloric Acid SCHEMBL6659919 0.75 ALDH1A1 (0.51) POLBALDH1A1TSHRCYP1A2LMNA
Hydrochloric Acid SCHEMBL6659351 0.74 SIGMAR1 (0.49) FAAHSIGMAR1HRH3
SCHEMBL27856022 0.73 POLB (0.70) POLBPKMALDH1A1FAAHSMN1; SMN2
SCHEMBL19002261 0.72 POLB (0.73) POLBPKMALDH1A1FAAHSMN1; SMN2
SCHEMBL19049377 0.72 HRH3 (0.71) POLBPKMALDH1A1FAAHSMN1; SMN2
SCHEMBL6630360 0.72 SIGMAR1 (0.69) POLBPKMALDH1A1FAAHSMN1; SMN2
SCHEMBL20804352 0.70 SIGMAR1 (0.85) POLBPKMALDH1A1SMN1; SMN2SIGMAR1
SCHEMBL1043952 0.70 SIGMAR1 (0.85) POLBPKMALDH1A1SMN1; SMN2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441728-A2 MODULATORS OF THE CHOLESTEROL BIOSYNTHETIC PATHWAY Vertex Pharmaceuticals Incorporated (US) 2004-08-04 EP disclosed
WO-2003037338-A2 MODULATORS OF THE CHOLESTEROL BIOSYNTHETIC PATHWAY VERTEX PHARMACEUTICALS INCORPORATED (US) 2003-05-08 WO disclosed
EP-1257544-A2 PIPERAZINE AND PIPERIDINE DERIVATIVES FOR TREATMENT OR PREVENTION OF NEURONAL DAMAGE Vertex Pharmaceuticals Incorporated (US) 2002-11-20 EP disclosed
WO-2001058891-A2 PIPERAZINE AND PIPERIDINE DERIVATIVES FOR TREATMENT OR PREVENTION OF NEURONAL DAMAGE VERTEX PHARMACEUTICALS INCORPORATED (US) 2001-08-16 WO disclosed