SCHEMBL6663415

SCHEMBL6663415

NNCNc1cccc(SCc2ccc(-c3ccccc3)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.45
GRK2 P25098 1/20 0.45
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
KDM4E B2RXH2 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
FFAR1 O14842 1/20 0.39
SLC6A4 P31645 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HAO1 Q9UJM8 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
DAO P14920 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679870 0.87 MAPT (0.43) ROCK2GRK2MAPTHTTMEN1
SCHEMBL6663788 0.81 MAOB (0.48) MAPTMEN1KMT2AKDM4EMAOA
SCHEMBL6154721 0.79 IDO1 (0.46) MAPTHTTMEN1KMT2AKDM4E
SCHEMBL6154708 0.76 MAOA (0.50) MEN1KMT2ATAAR1SLC6A4CYP3A4
Ammonia Solution, Strong SCHEMBL6679866 0.75 MAOA (0.48) MEN1KMT2ATAAR1SLC6A4CYP3A4
SCHEMBL6154702 0.74 MAOA (0.42) MAPTHTTMEN1KMT2AKDM4E
SCHEMBL19973146 0.73 MAOA (0.51) SLC6A4CYP3A4HAO1MAOAMAOB
SCHEMBL1323274 0.68 MAOB (0.54) ROCK2GRK2MAPTHTTMEN1
SCHEMBL6076179 0.68 MAOA (0.60) MEN1KMT2ATAAR1SLC6A4CYP3A4
SCHEMBL5391138 0.67 ALDH1A1 (0.62) MAPTMEN1KMT2AKDM4ETAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed