SCHEMBL6664491

SCHEMBL6664491

COc1ccc2nc(C(N)=O)cc(C3CC(C(=O)O)CCN3CCc3ccc4oc(=O)[nH]c4c3)c2n1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A3 Q01959 2/20 0.35
PDE10A Q9Y233 2/20 0.33
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 2/20 0.30
MCHR2 Q969V1 1/20 0.30
MCHR1 Q99705 1/20 0.30
GRM2 Q14416 1/20 0.30
TP53 P04637 1/20 0.30
PADI4 Q9UM07 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666166 0.84 KCNH2 (0.39) HTR1ASLC6A4KCNH2
SCHEMBL6661599 0.79 SLC2A1 (0.36) KCNH2
SCHEMBL6669040 0.78 KCNH2 (0.45) KCNH2
SCHEMBL6664492 0.76 KCNH2 (0.41) HTR1ASLC6A2SLC6A3KCNH2
SCHEMBL6669762 0.73 ALDH1A1 (0.40) KCNH2KMT2A
SCHEMBL14573151 0.72 KCNH2 (0.47) KCNH2
SCHEMBL5657364 0.68 HTR1A (0.49) HTR1ASLC6A2SLC6A3SLC6A4KCNH2
SCHEMBL5765881 0.67 KCNH2 (0.45) KCNH2
SCHEMBL6666267 0.66 MEN1 (0.37) HTR1AKMT2A
SCHEMBL6667354 0.63 KCNH2 (0.44) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392686-A1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2004-03-03 EP claimed
WO-2002096907-A1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-05 WO claimed