SCHEMBL6661599

SCHEMBL6661599

COc1ccc2nc(C(N)=O)cc(C3CC(C(=O)O)CCN3CCc3nc4c(F)cccc4[nH]3)c2n1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.36
SLC40A1 Q9NP59 4/20 0.33
KCNH2 Q12809 3/20 0.33
PARP1 P09874 4/20 0.33
TNKS O95271 6/20 0.32
TNKS2 Q9H2K2 6/20 0.32
PARP2 Q9UGN5 2/20 0.32
RORC P51449 3/20 0.31
REN P00797 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664491 0.79 HTR1A (0.35) KCNH2
SCHEMBL6666166 0.78 KCNH2 (0.39) KCNH2
SCHEMBL6669040 0.77 KCNH2 (0.45) KCNH2
SCHEMBL6661601 0.74 KCNH2 (0.45) SLC2A1SLC40A1KCNH2
SCHEMBL6669762 0.72 ALDH1A1 (0.40) KCNH2
SCHEMBL14573148 0.70 KCNH2 (0.47) SLC2A1SLC40A1KCNH2
SCHEMBL5657093 0.70 CHRNA7 (0.47) SLC40A1PARP1PARP2
SCHEMBL5765657 0.65 KCNH2 (0.47) SLC2A1SLC40A1KCNH2
SCHEMBL5656451 0.64 KDM4E (0.53) SLC40A1
SCHEMBL14573161 0.63 SLC40A1 (0.40) SLC2A1SLC40A1KCNH2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392686-A1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2004-03-03 EP claimed
WO-2002096907-A1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-05 WO claimed