SCHEMBL6664501

SCHEMBL6664501

CC(c1ccc(F)cc1)(c1ccc(F)cc1)N1CCN(C(=O)[C@@H]2CCCCN2CC2CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.41
CNR2 P34972 3/20 0.41
WNT3 P56703 1/20 0.41
SFRP1 Q8N474 1/20 0.41
LMNA P02545 2/20 0.38
MAPT P10636 1/20 0.38
MCHR1 Q99705 4/20 0.37
NPBWR1 P48145 3/20 0.37
SIGMAR1 Q99720 2/20 0.37
HRH3 Q9Y5N1 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7521716 0.87 ALDH1A1 (0.50) WNT3SFRP1MCHR1NPBWR1KDM4E
SCHEMBL6904670 0.78 DPP8 (0.49) CNR1CNR2LMNAMAPTALDH1A1
SCHEMBL6664503 0.77 MEN1 (0.42) WNT3SFRP1LMNAMCHR1NPBWR1
Hydrochloric Acid SCHEMBL6655911 0.70 KMT2A (0.50) KDM4EALDH1A1
Hydrochloric Acid SCHEMBL6906622 0.70 KMT2A (0.50) KDM4EALDH1A1
SCHEMBL6663657 0.69 HSD11B1 (0.55) LMNAKDM4EALDH1A1
SCHEMBL6908168 0.69 L3MBTL1 (0.50)
SCHEMBL6663653 0.69 HSD11B1 (0.55) LMNAKDM4EALDH1A1
SCHEMBL6659429 0.69 L3MBTL1 (0.50)
SCHEMBL6902204 0.68 DPP8 (0.50) CNR1CNR2LMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441728-A2 MODULATORS OF THE CHOLESTEROL BIOSYNTHETIC PATHWAY Vertex Pharmaceuticals Incorporated (US) 2004-08-04 EP disclosed
WO-2003037338-A2 MODULATORS OF THE CHOLESTEROL BIOSYNTHETIC PATHWAY VERTEX PHARMACEUTICALS INCORPORATED (US) 2003-05-08 WO disclosed