SCHEMBL6668575

SCHEMBL6668575

C=CC(=O)NCc1ccsc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 1/20 0.56
GRM5 P41594 2/20 0.47
HDAC6 Q9UBN7 2/20 0.45
HDAC8 Q9BY41 1/20 0.45
THRB P10828 1/20 0.41
HPGD P15428 1/20 0.41
ALDH1A1 P00352 4/20 0.41
TDP1 Q9NUW8 2/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
KDM4C Q9H3R0 1/20 0.40
NAMPT P43490 1/20 0.40
NPC1 O15118 1/20 0.39
LMNA P02545 2/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
HDAC1 Q13547 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18415493 0.84 HDAC6 (0.50) GRM5HDAC6HDAC8THRBHPGD
SCHEMBL18415486 0.80 GRM5 (0.53) GRM5HDAC6HDAC8THRBHPGD
SCHEMBL732934 0.79 TGM2 (0.81) TGM2ALDH1A1TDP1TSHRMAPK1
Thiophene SCHEMBL28891798 0.77 TGM2 (0.57) TGM2HPGDALDH1A1TSHRLMNA
SCHEMBL9430237 0.77 GRM5 (0.50) GRM5HDAC6HDAC8THRBHPGD
SCHEMBL26181255 0.75 TGM2 (0.63) TGM2ALDH1A1TDP1TSHRMAPK1
SCHEMBL6720904 0.75 GRM5 (0.52) GRM5HDAC6HDAC8THRBHPGD
SCHEMBL9480522 0.75 THRB (0.49) GRM5HDAC6HDAC8THRBHPGD
SCHEMBL12990668 0.75 GRM5 (0.46) GRM5HDAC6HDAC8THRBHPGD
SCHEMBL40744 0.74 TGM2 (0.68) TGM2HPGDALDH1A1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1226138-B1 FAB I INHIBITORS AFFINIUM PHARM INC (CA) 2004-12-29 EP disclosed