SCHEMBL6669755

SCHEMBL6669755

Cc1oc2ccc(NC(=O)C3CC3)nc2c1CCN(C)Cc1ccnc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 1/20 0.45
JAK2 O60674 6/20 0.38
TYK2 P29597 6/20 0.38
ALDH1A1 P00352 2/20 0.37
TSHR P16473 2/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
GSK3B P49841 3/20 0.33
HIF1A Q16665 1/20 0.33
JAK1 P23458 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546895 0.85 MEN1 (0.43) ALDH1A1HTTKMT2ANPC1RAB9A
SCHEMBL6672030 0.78 HTR1F (0.46) HTR1FALDH1A1TSHRCYP1A2CYP2D6
SCHEMBL8180841 0.74 HTR1F (0.44) HTR1FALDH1A1KMT2AMTNR1AMTNR1B
SCHEMBL8551076 0.70 CNR2 (0.41) ALDH1A1TSHRHTTKMT2ANPC1
SCHEMBL8550531 0.70 EGFR (0.42) ALDH1A1TSHRNPC1RAB9AHPGD
SCHEMBL8550370 0.69 KDM4E (0.41) ALDH1A1HTTKMT2ANPC1RAB9A
SCHEMBL6641025 0.68 HTR1F (0.71) HTR1FMTNR1AMTNR1B
SCHEMBL6641956 0.68 HTR1F (0.81) HTR1FALDH1A1CYP1A2CYP2D6KMT2A
SCHEMBL6668295 0.65 HTR1F (0.44) HTR1FALDH1A1KMT2ANPC1RAB9A
SCHEMBL7145980 0.63 HTR1F (0.43) HTR1FALDH1A1CYP1A2KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696439-B1 HETEROCYCLIC IMINES SUCH AS 2-METHYL-3-(2-(N',N'-DIETHYLAMINO) ETHYL)-5-(4-PROPANESULFONYLBENZAMIDE)FURO(3,2-B)PYRIDINE, HYDROCHLORIDE, USED AS SEROTONIN RECEPTOR ANTAGONISTS FOR PROPHYLAXIS OF HEADACHES ELI LILLY AND COMPANY 2004-02-24 US disclosed
EP-1155020-B1 FURO[3,2-B]PYRIDINES AS 5-HT1F AGONISTS LILLY CO ELI (US) 2004-02-04 EP disclosed