SCHEMBL6672030

SCHEMBL6672030

Cc1oc2ccc(NC(=O)C3CCCCCC3)nc2c1CCN(C)Cc1nccs1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 3/20 0.46
RAB9A P51151 6/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 3/20 0.37
ALDH1A1 P00352 4/20 0.37
TSHR P16473 3/20 0.37
KMT2A Q03164 3/20 0.37
CYP1A2 P05177 2/20 0.37
HTT P42858 2/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTR1A P08908 2/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 2/20 0.35
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553305 0.85 SMN1; SMN2 (0.42) RAB9ASMN1; SMN2NPC1ALDH1A1TSHR
SCHEMBL6667543 0.79 HTR1F (0.44) HTR1FRAB9ANPC1ALDH1A1TSHR
SCHEMBL6669755 0.78 HTR1F (0.45) HTR1FRAB9ANPC1ALDH1A1TSHR
SCHEMBL8553336 0.74 SMN1; SMN2 (0.40) RAB9ASMN1; SMN2NPC1ALDH1A1TSHR
SCHEMBL8180418 0.74 HTR1F (0.43) HTR1FRAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL6641025 0.69 HTR1F (0.71) HTR1FL3MBTL1KDM4E
SCHEMBL8550329 0.66 KDM4E (0.40) SMN1; SMN2ALDH1A1KDM4E
SCHEMBL6668295 0.65 HTR1F (0.44) HTR1FRAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL6641956 0.65 HTR1F (0.81) HTR1FRAB9ANPC1ALDH1A1KMT2A
Acetic Acid SCHEMBL8548884 0.65 JAK2 (0.39) RAB9ASMN1; SMN2NPC1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696439-B1 HETEROCYCLIC IMINES SUCH AS 2-METHYL-3-(2-(N',N'-DIETHYLAMINO) ETHYL)-5-(4-PROPANESULFONYLBENZAMIDE)FURO(3,2-B)PYRIDINE, HYDROCHLORIDE, USED AS SEROTONIN RECEPTOR ANTAGONISTS FOR PROPHYLAXIS OF HEADACHES ELI LILLY AND COMPANY 2004-02-24 US disclosed
EP-1155020-B1 FURO[3,2-B]PYRIDINES AS 5-HT1F AGONISTS LILLY CO ELI (US) 2004-02-04 EP disclosed