SCHEMBL6670152

SCHEMBL6670152

CC(C)(C)CC(=O)N1CCc2ccccc2C1CCN1CCC(c2cccc3c2OCC3)CC1.COc1cc2c(cc1OC)C(CCN1CCC(O)(c3ccc(Cl)c(C(F)(F)F)c3)CC1)N(C(=O)CC(C)(C)C)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 10/20 0.41
OPRL1 P41146 7/20 0.41
SCN1A P35498 1/20 0.39
SCN2A Q99250 1/20 0.39
SCN3A Q9NY46 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
OPRD1 P41143 4/20 0.37
OPRK1 P41145 4/20 0.37
HTR1A P08908 3/20 0.37
DRD2 P14416 3/20 0.37
DRD4 P21917 3/20 0.37
HTR1D P28221 3/20 0.37
HTR2A P28223 3/20 0.37
HTR2C P28335 3/20 0.37
HTR7 P34969 3/20 0.37
DRD1 P21728 2/20 0.37
DRD5 P21918 2/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
DRD3 P35462 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4839599 0.87 OPRM1 (0.48) OPRM1OPRL1SCN1ASCN2ASCN3A
SCHEMBL4839787 0.80 HTR2A (0.47) DRD2HTR2ADRD3
SCHEMBL4838194 0.77 MTNR1B (0.53) OPRM1OPRL1SCN1ASCN2ASCN3A
SCHEMBL4832883 0.77 OPRM1 (0.48) OPRM1OPRL1SCN1ASCN2ASCN3A
SCHEMBL4839076 0.69 DRD2 (0.51) OPRD1DRD2DRD4MEN1KMT2A
SCHEMBL4837162 0.68 DRD2 (0.40) HTR1ADRD2HTR1DHTR2ADRD3
SCHEMBL6668370 0.68 MTNR1B (0.43) MTNR1BMEN1KMT2A
SCHEMBL4838758 0.68 MCHR1 (0.46) DRD2DRD4DRD3MEN1KMT2A
SCHEMBL4836909 0.67 NPSR1 (0.49) HTR1ADRD2HTR1DHTR2ADRD3
SCHEMBL4839490 0.67 HTR2A (0.47) HTR1ADRD2DRD4HTR1DHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458714-A1 3,4-DIHYDRO-1H-ISOQUINOLOIN-2-YL-DERIVATIVES H. Lundbeck A/S (DK) 2004-09-22 EP claimed
WO-2003051869-A1 3,4-DIHYDRO-1H-ISOQUINOLOIN-2-YL-DERIVATIVES H. LUNDBECK A/S (DK) 2003-06-26 WO claimed