SCHEMBL6671176

SCHEMBL6671176

Cc1cccc(C(=O)Cc2ccnc3cc(F)ccc23)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
POLB P06746 1/20 0.40
KMT2A Q03164 1/20 0.40
ACVR1 Q04771 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
FERMT2 Q96AC1 1/20 0.39
P2RX7 Q99572 1/20 0.39
GRM5 P41594 4/20 0.38
GBA1 P04062 2/20 0.38
TP53 P04637 1/20 0.36
PDGFRB P09619 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CDK8 P49336 1/20 0.35
CLK2 P49760 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
AAK1 Q2M2I8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24322279 0.92 CDK8 (0.39) NPC1RAB9ASMN1; SMN2POLBKMT2A
SCHEMBL5234890 0.88 P2RX7 (0.39) NPC1RAB9ASMN1; SMN2POLBKMT2A
SCHEMBL5231489 0.86 PRNP (0.45) SMN1; SMN2POLBKMT2AACVR1CLK4
SCHEMBL4490632 0.86 P2RX7 (0.39) NPC1RAB9ASMN1; SMN2POLBKMT2A
SCHEMBL5236990 0.85 GSK3A (0.44) ACVR1CLK4P2RX7CLK2DYRK1B
SCHEMBL5235795 0.84 KDR (0.45) NPC1RAB9AACVR1CLK4FERMT2
SCHEMBL5235225 0.84 CYP1A2 (0.49) RAB9ASMN1; SMN2P2RX7GRM5ALDH1A1
SCHEMBL29959459 0.84 CYP1A2 (0.49) RAB9ASMN1; SMN2P2RX7GRM5ALDH1A1
SCHEMBL5238328 0.83 THRB (0.44) NPC1RAB9ASMN1; SMN2KMT2AP2RX7
SCHEMBL5231308 0.81 SRC (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004026302-A1 METHODS OF INHIBITING TGF BETA WITH SUBSTITUTED PYRAZOLES ELI LILLY AND COMPANY (US) 2004-04-01 WO disclosed