SCHEMBL6671955

SCHEMBL6671955

Cc1ccc(C(=O)NC(N)(C(=NC#N)Nc2ccccc2)C(Cl)(Cl)Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
MAPT P10636 3/20 0.42
TDP1 Q9NUW8 1/20 0.40
ALDH1A1 P00352 6/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
NTSR1 P30989 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 3/20 0.38
TNIK Q9UKE5 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
ABCC9 O60706 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6611894 0.87 KCNJ11 (0.40) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL6668769 0.82 NAMPT (0.51) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL6611441 0.82 NAMPT (0.51) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL6612062 0.79 NPC1 (0.41) NPC1RAB9AMAPTALDH1A1MEN1
SCHEMBL6614765 0.79 NAMPT (0.55) NPC1RAB9ASMN1; SMN2ABCC9KCNJ11
SCHEMBL6609354 0.73 ABCC9 (0.53) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL4681399 0.72 LMNA (0.48) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL4681401 0.72 LMNA (0.48) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL6612688 0.69 CYP11B1 (0.54) NPC1RAB9ASMN1; SMN2ABCC9KCNJ11
SCHEMBL6669216 0.69 RAB9A (0.47) NPC1RAB9ASMN1; SMN2ABCC9KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392655-A2 POTASSIUM CHANNEL OPENERS Abbott Laboratories (US) 2004-03-03 EP disclosed
WO-2002062762-A2 POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2002-08-15 WO disclosed