SCHEMBL6675013

SCHEMBL6675013

CCc1cc(N=C(NO)N2CCN(c3ccccc3SC)CC2)c(OC)nc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.35
HTR1A P08908 4/20 0.35
DRD4 P21917 2/20 0.34
DRD3 P35462 1/20 0.34
PKM P14618 1/20 0.34
HTT P42858 2/20 0.34
HTR2A P28223 1/20 0.34
MEN1 O00255 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 2/20 0.33
POLB P06746 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678795 0.91 PKM (0.37) PKMHTTKMT2ARAB9AGAA
SCHEMBL6678709 0.90 DRD2 (0.35) DRD2HTR1ADRD4DRD3HTT
SCHEMBL6675058 0.89 KMT2A (0.34) DRD2HTR1ADRD4HTTMEN1
SCHEMBL6673628 0.88 PKM (0.46) PKMHTTCYP2C19KMT2ARAB9A
SCHEMBL6675441 0.87 RAB9A (0.36) DRD2HTR1ADRD4DRD3HTT
SCHEMBL6673642 0.86 THRB (0.37) DRD2HTR1ADRD4DRD3HTT
SCHEMBL6676096 0.86 KMT2A (0.32) DRD2HTR1ADRD4HTTMEN1
SCHEMBL6674452 0.85 HSD17B10 (0.42) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL6673300 0.84 MEN1 (0.31) DRD2HTR1ADRD4HTTMEN1
SCHEMBL6678502 0.84 DRD4 (0.33) DRD2HTR1ADRD4HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1424072-A1 N'-(pyridin-3-yl)-(4-phenylpiperazin-1-yl)-carboxyimidamide and -iminothiolate derivatives for the treatment of tumors Samjin Pharmaceutical Co., Ltd. (KR) 2004-06-02 EP disclosed
US-6683184-B2 ANTITUMOR AGENTS SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2004-01-27 US disclosed