SCHEMBL6676085

SCHEMBL6676085

CC#CCOc1ccc(S(=O)(=O)N(CCN2CCOCC2)[C@H](C)CSC(C)=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 15/20 0.46
MMP13 P45452 11/20 0.46
MMP2 P08253 8/20 0.46
MMP1 P03956 7/20 0.44
MMP9 P14780 7/20 0.44
MMP14 P50281 2/20 0.43
MMP3 P08254 1/20 0.43
BMP1 P13497 1/20 0.42
MMP7 P09237 2/20 0.41
MMP8 P22894 2/20 0.41
ADAM10 O14672 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675605 0.88 ADAM17 (0.47) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6330947 0.87 ALDH1A1 (0.48) MMP13MMP2MMP3BMP1HDAC3
SCHEMBL3944994 0.86 ADAM17 (0.50) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6504827 0.83 MMP13 (0.55) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6508689 0.82 MMP13 (0.53) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL3943732 0.81 MMP13 (0.66) ADAM17MMP13MMP2MMP1MMP9
Hydrochloric Acid SCHEMBL6498659 0.81 MMP13 (0.65) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6625710 0.81 MMP13 (0.46) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL3950424 0.80 ADAM17 (0.46) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6325041 0.79 HRH3 (0.47) MMP13MMP1MMP9HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1149074-B1 ACETYLENIC SULFONAMIDE THIOL TACE INHIBITORS WYETH CORP (US) 2004-10-20 EP disclosed
US-6313123-B1 FOR THERAPY OF RHEUMATOID ARTHRITIS, OSTEOARTHRITIS, SEPSIS, AIDS, ULCERATIVE COLITIS, MULTIPLE SCLEROSIS, CROHN'S DISEASE AND DEGENERATIVE CARTILAGE LOSS AMERICAN CYANAMID COMPANY 2001-11-06 US disclosed
EP-1149074-A1 ACETYLENIC SULFONAMIDE THIOL TACE INHIBITORS American Cyanamid Company (US) 2001-10-31 EP disclosed
WO-2000044716-A1 ACETYLENIC SULFONAMIDE THIOL TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO disclosed