SCHEMBL6676115

SCHEMBL6676115

CCNC(=NC(=O)OC(C)(C)C)Nc1ccc(CCNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.53
CA2 P00918 6/20 0.44
CA1 P00915 4/20 0.44
CYP17A1 P05093 1/20 0.42
PTPRB P23467 1/20 0.40
CNR1 P21554 1/20 0.40
PTGER4 P35408 1/20 0.39
PTPN11 Q06124 1/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DRD2 P14416 1/20 0.39
CTSK P43235 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
GLA P06280 1/20 0.38
KMT2A Q03164 1/20 0.38
IGF1R P08069 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6677735 0.88 NAMPT (0.53) NAMPTCA2CA1CYP17A1CNR1
SCHEMBL6687612 0.84 IDO1 (0.43) NAMPTCA2CA1CNR1MAPT
SCHEMBL6676262 0.84 PTGER4 (0.41) NAMPTCA2CA1PTPRBCNR1
SCHEMBL6681072 0.83 NQO2 (0.40) NAMPTCA2CA1PTPN11MAPT
SCHEMBL6675282 0.83 NAMPT (0.40) NAMPTCA2CA1PTPRBPTGER4
SCHEMBL7248121 0.83 MEN1 (0.41) NAMPTCA2CA1CYP17A1PTGER4
SCHEMBL6689914 0.82 ALDH1A1 (0.41) NAMPTCNR1DRD2KMT2A
SCHEMBL6681999 0.82 MAPT (0.45) NAMPTCA2CA1MAPTNPSR1
SCHEMBL3787072 0.81 CYP17A1 (0.47) NAMPTCA2CA1CYP17A1PTPN11
SCHEMBL13017220 0.81 CYP17A1 (0.47) NAMPTCA2CA1CYP17A1PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed