SCHEMBL6676832

SCHEMBL6676832

NCc1ccc(NC(N)=NC2CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 2/20 0.41
GRIN3B O60391 2/20 0.41
GRIN1 Q05586 2/20 0.41
GRIN2A Q12879 2/20 0.41
GRIN2B Q13224 2/20 0.41
GRIN2C Q14957 2/20 0.41
GRIN3A Q8TCU5 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
CXCR3 P49682 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6674864 0.84 SIGMAR1 (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL30182461 0.72 KMT2A (0.74) MEN1LMNAKMT2A
SCHEMBL30182449 0.72 KMT2A (0.74) MEN1LMNAKMT2A
SCHEMBL2579208 0.72 KMT2A (0.74) MEN1LMNAKMT2A
SCHEMBL6676200 0.69 LOXL2 (0.44) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL327252 0.69 LOXL2 (0.54) PLAUKLKB1PLGPLATPRSS1
SCHEMBL8530522 0.69 PEPD (0.59) MEN1LMNAKMT2APLAUKLKB1
SCHEMBL6833494 0.69 ALDH1A1 (0.56) KMT2ATP53CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7443406 0.67 LOXL2 (0.52) PLAUKLKB1PLGPLATPRSS1
SCHEMBL6676828 0.67 PRSS1 (0.40) MEN1LMNAKMT2APLAUKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP claimed
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed