SCHEMBL6676955

SCHEMBL6676955

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(O)c(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.43
HDAC1 Q13547 1/20 0.40
ANO1 Q5XXA6 1/20 0.40
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
PTPN11 Q06124 1/20 0.38
ACHE P22303 1/20 0.37
BACE1 P56817 1/20 0.37
NAMPT P43490 1/20 0.37
NR1H4 Q96RI1 2/20 0.37
KDM4A O75164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678684 0.87 ALDH1A1 (0.43) PTPN11NAMPTNR1H4
SCHEMBL6674829 0.86 PTPN1 (0.38) PTPN11NAMPTNR1H4KDM4A
SCHEMBL6676957 0.82 EGFR (0.43) EGFRHDAC1ANO1CA1CA2
SCHEMBL6680473 0.81 CYP2C9 (0.42) HDAC1NAMPT
SCHEMBL6681934 0.79 ALDH1A1 (0.42) NAMPT
SCHEMBL6687607 0.79 IDO1 (0.44) EGFRANO1CA1CA2PTPN11
SCHEMBL6675974 0.79 CA1 (0.36) CA1CA2PTPN11NR1H4
SCHEMBL6681071 0.78 NQO2 (0.41) EGFRHDAC1CA1CA2PTPN11
SCHEMBL6679938 0.77 NR1H4 (0.36) CA1CA2PTPN11NR1H4
SCHEMBL7243630 0.77 ALDH1A1 (0.42) CA1CA2NAMPTNR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed