SCHEMBL6677982

SCHEMBL6677982

C[C@H](Cc1ccc(S(=O)(=O)c2cccc(-c3cccc(C(=O)O)c3)c2)cc1)NC(=O)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.40
KCNH2 Q12809 1/20 0.40
MME P08473 1/20 0.40
MMEL1 Q495T6 1/20 0.40
PFKFB3 Q16875 1/20 0.39
CDK2 P24941 1/20 0.39
F2 P00734 3/20 0.38
TMPRSS6 Q8IU80 2/20 0.38
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
ABCC9 O60706 3/20 0.38
ABCC8 Q09428 3/20 0.38
KCNJ11 Q14654 3/20 0.38
KCNJ8 Q15842 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ACACB O00763 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805111 0.88 ACACB (0.48) ESR1KCNH2ACACB
SCHEMBL6677082 0.85 ACACB (0.50) ESR1KCNH2L3MBTL1ACACB
SCHEMBL6676495 0.84 ALDH1A1 (0.47) L3MBTL1ACACB
SCHEMBL6805115 0.84 APAF1 (0.37) ESR1KCNH2MMEMMEL1CDK2
SCHEMBL6540275 0.83 ABCC9 (0.55) ESR1KCNH2ABCC9ABCC8KCNJ11
SCHEMBL6805113 0.82 SYK (0.43) ESR1KCNH2CDK2ITGB1ITGA4
SCHEMBL6540336 0.81 ACACB (0.52) ESR1KCNH2ABCC9ABCC8KCNJ11
SCHEMBL6809925 0.81 CNR1 (0.38) ESR1KCNH2MMEMMEL1ABCC9
SCHEMBL6799811 0.81 ABCC9 (0.45) ESR1KCNH2ABCC9ABCC8KCNJ11
SCHEMBL6540797 0.81 ABCC9 (0.45) ESR1KCNH2ABCC9ABCC8KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004045610-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD (JP) 2004-06-03 WO disclosed