SCHEMBL6678068

SCHEMBL6678068

CC(C)(C)OC(=O)N(Cc1cccc(N)c1Cl)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.36
SLC6A4 P31645 2/20 0.34
GRM2 Q14416 1/20 0.34
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
CPB2 Q96IY4 1/20 0.32
AAK1 Q2M2I8 1/20 0.32
HTR2C P28335 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
MT-CO2 P00403 1/20 0.32
AKT1 P31749 2/20 0.32
NQO2 P16083 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ESR1 P03372 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25399427 0.85 GRM2 (0.35) GRM2AAK1HDAC3HDAC1HDAC2
SCHEMBL6677666 0.84 ESR1 (0.42) GRM2AAK1HDAC3HDAC1HDAC2
SCHEMBL6677867 0.82 KDM4E (0.36) GRM2L3MBTL1
SCHEMBL7872408 0.80 HDAC1 (0.34) GRM2CPB2HDAC3HDAC1HDAC2
SCHEMBL7880189 0.79 AAK1 (0.34) GRM2AAK1ESR1KCNH2
SCHEMBL6679943 0.79 NR1D1 (0.40) NR1H3
SCHEMBL13656744 0.79 NR1D1 (0.40) GRM2HDAC3HDAC1HDAC2NCOR2
SCHEMBL27402130 0.79 KDM4E (0.39) SLC6A4KCNH2
SCHEMBL1626936 0.78 TSHR (0.40) GRM2HDAC3HDAC1HDAC2NCOR2
SCHEMBL6678098 0.78 GPR35 (0.39) RENL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed