SCHEMBL7872408

SCHEMBL7872408

CCOc1c(N)cccc1CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 3/20 0.33
CPB2 Q96IY4 4/20 0.33
GRM2 Q14416 1/20 0.32
AKT1 P31749 2/20 0.32
NPC1 O15118 1/20 0.32
USP2 O75604 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
CREBBP Q92793 1/20 0.31
CHEK1 O14757 1/20 0.31
GABRA1 P14867 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7880112 0.90 HDAC3 (0.33) HDAC1HDAC3HDAC2NCOR2ALDH1A1
SCHEMBL6677867 0.86 KDM4E (0.36) ALDH1A1TSHRHSD17B10GRM2NPC1
SCHEMBL7880189 0.83 AAK1 (0.34) TSHRGRM2
SCHEMBL25399427 0.82 GRM2 (0.35) HDAC1HDAC3HDAC2NCOR2ALDH1A1
SCHEMBL6677666 0.81 ESR1 (0.42) HDAC1HDAC3HDAC2NCOR2ALDH1A1
SCHEMBL7876745 0.80 ALDH1A1 (0.42) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL6678068 0.80 REN (0.36) HDAC1HDAC3HDAC2NCOR2CPB2
SCHEMBL13656744 0.75 NR1D1 (0.40) HDAC1HDAC3HDAC2NCOR2TSHR
SCHEMBL1626936 0.75 TSHR (0.40) HDAC1HDAC3HDAC2NCOR2ALDH1A1
SCHEMBL26256957 0.74 AAK1 (0.33) TSHRGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6331553-B1 INHIBITORS OF NITRIC OXIDE SYNTHASE; TREATING CEREBROVASCULAR DISEASES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-12-18 US disclosed
EP-0949242-A1 AROMATIC AMINE DERIVATIVES HAVING NOS INHIBITORY EFFECT Chugai Seiyaku Kabushiki Kaisha (JP) 1999-10-13 EP disclosed