SCHEMBL6679699

SCHEMBL6679699

Cc1cc(-c2ccccc2)c(C(=O)Nc2ccc(NCCc3cccc(N)n3)cc2)cc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.43
S1PR3 Q99500 9/20 0.43
OPRL1 P41146 1/20 0.39
TRPV4 Q9HBA0 1/20 0.39
PTGS1 P23219 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678979 0.89 PDGFRB (0.43) S1PR1S1PR3PTGS1
SCHEMBL6677053 0.89 ITGB1 (0.44) S1PR1S1PR3OPRL1
SCHEMBL6685612 0.87 S1PR1 (0.46) S1PR1S1PR3
SCHEMBL6677401 0.85 SORT1 (0.39) S1PR1S1PR3TRPV4
SCHEMBL7083682 0.84 CA12 (0.45) TRPV4PTGS1
SCHEMBL6499114 0.84 HDAC7 (0.47) OPRL1
SCHEMBL6489781 0.84 L3MBTL1 (0.47) OPRL1
SCHEMBL6683660 0.81 S1PR1 (0.48) S1PR1S1PR3PTGS1
SCHEMBL6638338 0.81 S1PR1 (0.43) S1PR1S1PR3
SCHEMBL7081444 0.81 TP53 (0.43) OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1472226-A1 HETEROCYCLIC AMIDE COMPOUNDS AS APOLIPOPROTEIN B INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-03 EP disclosed
WO-2003045921-A1 HETEROCYCLIC AMIDE COMPOUNDS AS APOLIPOPROTEIN B INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-06-05 WO disclosed