SCHEMBL6680366

SCHEMBL6680366

FC(F)(F)c1cc(B2OB(c3cc(C(F)(F)F)cc(C(F)(F)F)c3)OB(c3cc(C(F)(F)F)cc(C(F)(F)F)c3)O2)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.39
IDO1 P14902 2/20 0.35
ADRB1 P08588 1/20 0.32
MAPT P10636 1/20 0.31
RAPGEF4 Q8WZA2 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGAV P06756 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31
ALDH1A1 P00352 2/20 0.31
TSHR P16473 1/20 0.31
CES1 P23141 1/20 0.30
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6692161 0.79 CES2 (0.35) CES2IDO1ADRB1
SCHEMBL2432674 0.78 TSHR (0.47) CES2IDO1MAPTALDH1A1TSHR
SCHEMBL10379650 0.78 CES2 (0.39) CES2IDO1MAPTRXRARXRB
SCHEMBL5077943 0.76 LPL (0.43) CES2
SCHEMBL7784283 0.76 CES2 (0.33) CES2IDO1ITGB3ITGAV
SCHEMBL7859828 0.75 CES2 (0.44) CES2IDO1ALDH1A1TSHRCES1
SCHEMBL14227219 0.74 CES2 (0.32) CES2
SCHEMBL14227199 0.74 TSHR (0.38) CES2IDO1MAPTRXRARXRB
SCHEMBL440959 0.74 CES2 (0.58) CES2IDO1ADRB1MAPTRAPGEF4
SCHEMBL8587206 0.71 CES2 (0.33) CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137641-B1 PROCESS FOR PREPARING PYRIDAZIN-3-ON DERIVATIVES SUMITOMO CHEMICAL CO (JP) 2004-11-10 EP disclosed
US-6500951-B1 RING CLOSING A CARBOXYLIC ACID DERIVATIVE IN PRESENCE OF A NITROGEN CONTAINING AROMATIC COMPOUND AND A BORON COMPOUND; HIGH YIELD AND PURITY SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-12-31 US disclosed