SCHEMBL6681291

SCHEMBL6681291

CN(Cc1ccccc1)Cc1cccc(NC(N)=S)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
TP53 P04637 1/20 0.51
TYR P14679 1/20 0.51
TSHR P16473 1/20 0.51
TAS2R38 P59533 1/20 0.51
HSD17B10 Q99714 1/20 0.51
CYP1A2 P05177 1/20 0.51
KMT2A Q03164 3/20 0.49
ACHE P22303 5/20 0.48
ALOX5 P09917 1/20 0.48
BACE1 P56817 1/20 0.48
BCHE P06276 4/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
MEN1 O00255 2/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
PTGES O14684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3597276 0.86 CYP1A2 (0.56) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL27477068 0.82 KMT2A (0.49) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL6676464 0.81 SIGMAR1 (0.48) KMT2AACHEALOX5BACE1BCHE
Hydrochloric Acid SCHEMBL6679385 0.80 SIGMAR1 (0.49) ACHEALOX5BACE1BCHEMAOA
SCHEMBL3427115 0.80 ALDH1A1 (0.60) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL1887849 0.78 CYP1A2 (0.61) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL7238879 0.78 BACE1 (0.51) ALDH1A1CYP1A2KMT2ABACE1MEN1
SCHEMBL27552470 0.78 ALDH1A1 (0.44) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL7600769 0.77 ACHE (0.51) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL13338007 0.77 ALDH1A1 (0.56) ALDH1A1TP53TYRTSHRTAS2R38

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
CN-1310169-A Anils with nitric oxide synzyme inhibiting function SHUGAI SEIYAKU K K (JP) 2001-08-29 CN disclosed
CN-1172473-A Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 1998-02-04 CN disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed