SCHEMBL6681809

SCHEMBL6681809

Cn1cccc1CNCCCC(NC(=O)c1ccc(C(N)Cc2nccn2C)cc1)C(=O)O.NCc1cccc2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 2/20 0.39
TGM2 P21980 5/20 0.36
CASR P41180 2/20 0.36
CXCR4 P61073 1/20 0.33
C3AR1 Q16581 1/20 0.33
CCKBR P32239 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
DHFR P00374 1/20 0.32
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32
SLC40A1 Q9NP59 1/20 0.31
FNTA P49354 2/20 0.31
FNTB P49356 2/20 0.31
MC4R P32245 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6683363 0.94 FOLH1 (0.41) FOLH1TGM2CASRCXCR4C3AR1
SCHEMBL6681620 0.92 FOLH1 (0.43) FOLH1TGM2CASRC3AR1CCKBR
SCHEMBL6682711 0.89 CXCR4 (0.40) FOLH1TGM2CASRCXCR4HTT
SCHEMBL6688643 0.89 FOLH1 (0.38) FOLH1CASRC3AR1CCKBRHTT
SCHEMBL6685296 0.89 FOLH1 (0.38) FOLH1TGM2CASRCXCR4C3AR1
SCHEMBL6018574 0.82 CXCR4 (0.51) FOLH1TGM2CASRCXCR4DHFR
SCHEMBL6687483 0.81 CXCR4 (0.40) FOLH1TGM2CASRCXCR4DHFR
SCHEMBL6685578 0.81 FOLH1 (0.41) FOLH1CASRC3AR1CCKBR
SCHEMBL6018129 0.80 CXCR4 (0.51) FOLH1TGM2CASRCXCR4DHFR
SCHEMBL6690573 0.80 HDAC1 (0.40) FOLH1CASRCXCR4DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed