SCHEMBL6685296

SCHEMBL6685296

Cn1cccc1CNCCCC(NC(=O)c1ccc(C(N)Cc2nccs2)cc1)C(=O)O.NCc1cccc2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.38
CASR P41180 1/20 0.35
DHFR P00374 1/20 0.33
TGM2 P21980 4/20 0.32
MC4R P32245 1/20 0.32
CXCR4 P61073 1/20 0.32
C3AR1 Q16581 1/20 0.32
CCKBR P32239 1/20 0.32
FNTA P49354 2/20 0.31
FNTB P49356 2/20 0.31
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
PIN1 Q13526 1/20 0.30
KLKB1 P03952 1/20 0.30
KLK1 P06870 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6681620 0.90 FOLH1 (0.43) FOLH1CASRDHFRTGM2C3AR1
SCHEMBL6681809 0.89 FOLH1 (0.39) FOLH1CASRDHFRTGM2MC4R
SCHEMBL6688643 0.85 FOLH1 (0.38) FOLH1CASRC3AR1CCKBRKLK1
SCHEMBL6683363 0.83 FOLH1 (0.41) FOLH1CASRDHFRTGM2MC4R
SCHEMBL6018574 0.81 CXCR4 (0.51) FOLH1CASRDHFRTGM2CXCR4
SCHEMBL6682711 0.81 CXCR4 (0.40) FOLH1CASRDHFRTGM2CXCR4
SCHEMBL6687483 0.80 CXCR4 (0.40) FOLH1CASRDHFRTGM2CXCR4
SCHEMBL6017970 0.79 CXCR4 (0.41) FOLH1TGM2CXCR4CCKBR
SCHEMBL6687885 0.77 FOLH1 (0.41) FOLH1CASRTGM2
SCHEMBL6686504 0.77 CXCR4 (0.41) FOLH1CASRDHFRTGM2CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed