SCHEMBL6683363

SCHEMBL6683363

Cn1ccnc1CNCCCC(NC(=O)c1ccc(C(N)Cc2nccn2C)cc1)C(=O)O.NCc1cccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 2/20 0.41
CASR P41180 2/20 0.38
TGM2 P21980 5/20 0.37
C3AR1 Q16581 1/20 0.35
CXCR4 P61073 1/20 0.35
SLC40A1 Q9NP59 1/20 0.34
CCKBR P32239 1/20 0.34
DHFR P00374 1/20 0.34
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
FNTA P49354 2/20 0.32
FNTB P49356 2/20 0.32
MC4R P32245 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32
TPSAB1 Q15661 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6681809 0.94 FOLH1 (0.39) FOLH1CASRTGM2C3AR1CXCR4
SCHEMBL6682711 0.85 CXCR4 (0.40) FOLH1CASRTGM2CXCR4DHFR
SCHEMBL6018129 0.85 CXCR4 (0.51) FOLH1CASRTGM2CXCR4DHFR
SCHEMBL6685578 0.85 FOLH1 (0.41) FOLH1CASRC3AR1CCKBR
SCHEMBL6681620 0.85 FOLH1 (0.43) FOLH1CASRTGM2C3AR1CCKBR
SCHEMBL6690684 0.84 CXCR4 (0.40) FOLH1CASRTGM2CXCR4SLC40A1
SCHEMBL6690468 0.84 CXCR4 (0.40) FOLH1CASRTGM2CXCR4SLC40A1
SCHEMBL6694422 0.83 FOLH1 (0.47) FOLH1CASRTGM2SLC40A1FNTA
SCHEMBL6685296 0.83 FOLH1 (0.38) FOLH1CASRTGM2C3AR1CXCR4
SCHEMBL6688643 0.83 FOLH1 (0.38) FOLH1CASRC3AR1CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed