SCHEMBL6683040

SCHEMBL6683040

C=CCc1c(S(=O)(=O)O)ccc(C)c1CCCO

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CA2 P00918 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
BRD4 O60885 1/20 0.30
BRD2 P25440 1/20 0.30
BRD3 Q15059 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734598 0.81 MEN1 (0.35) ALDH1A1MEN1KMT2A
SCHEMBL2059594 0.79 POLB (0.33) MEN1KMT2A
SCHEMBL5412420 0.79 MEN1 (0.34) ALDH1A1NPSR1MEN1KMT2A
SCHEMBL28557476 0.78 MYC (0.37) ALDH1A1
SCHEMBL15968890 0.77 ALDH1A1 (0.35) ALDH1A1NPSR1CA2MEN1KMT2A
SCHEMBL2057642 0.77 MEN1 (0.30) MEN1KMT2A
SCHEMBL7758371 0.75 KDM4E (0.38) ALDH1A1NPSR1MEN1KMT2A
SCHEMBL8773429 0.74 POLB (0.33) ALDH1A1
SCHEMBL7597928 0.74 CASP1 (0.37) ALDH1A1NPSR1CA2MEN1KMT2A
SCHEMBL3744994 0.74 CTDSP1 (0.33) ALDH1A1NPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370547-B1 BENZOAXATHIEPIN DERIVATIVES AND THEIR USE AS MEDICINES PF MEDICAMENT (FR) 2004-09-15 EP disclosed
EP-1370547-A1 BENZOAXATHIEPIN DERIVATIVES AND THEIR USE AS MEDICINES PIERRE FABRE MEDICAMENT (FR) 2003-12-17 EP disclosed
WO-2002081464-A1 BENZOAXATHIEPIN DERIVATIVES AND THEIR USE AS MEDICINES PIERRE FABRE MEDICAMENT (FR) 2002-10-17 WO disclosed