SCHEMBL6684875

SCHEMBL6684875

O=C(NCc1ccc(F)cc1)c1ccc2c(c1)C(=O)C(Cc1ccc(F)c(Cl)c1)C(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.49
TP53 P04637 5/20 0.49
LMNA P02545 4/20 0.49
CNR1 P21554 1/20 0.45
POLB P06746 3/20 0.44
PPARG P37231 1/20 0.43
RXFP1 Q9HBX9 2/20 0.42
THRB P10828 1/20 0.42
WDR5 P61964 1/20 0.41
PTGER4 P35408 2/20 0.39
PTGER2 P43116 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678534 0.94 MAPT (0.48) MAPTTP53LMNACNR1POLB
SCHEMBL6680500 0.93 MAPT (0.47) MAPTTP53LMNACNR1POLB
SCHEMBL6684559 0.92 MAPT (0.53) MAPTTP53LMNACNR1POLB
SCHEMBL6683273 0.92 MAPT (0.49) MAPTTP53LMNACNR1POLB
SCHEMBL6682598 0.90 MAPT (0.51) MAPTTP53LMNAPOLBWDR5
SCHEMBL6679778 0.90 MAPT (0.47) MAPTTP53LMNACNR1POLB
SCHEMBL6681366 0.87 MAPT (0.56) MAPTTP53LMNACNR1POLB
SCHEMBL6664864 0.84 MAPT (0.47) MAPTTP53LMNACNR1POLB
SCHEMBL6666007 0.84 TRPV1 (0.39)
SCHEMBL6685985 0.83 MAPT (0.51) MAPTTP53LMNAPOLBWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors HICKS JAMES LESTER (US) 2004-03-04 US disclosed
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors MMP13, MMP26, MMP9 MAPT 2365/4885TP53 4473/4885LMNA 2566/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.