SCHEMBL6686940

SCHEMBL6686940

O=C(NCC(C(=O)NCCNc1ccc(OC(F)(F)F)cc1)C1CCCCC1)c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSS P25774 14/20 0.56
CTSL P07711 10/20 0.50
CTSK P43235 7/20 0.50
MAPK14 Q16539 1/20 0.47
TRPV1 Q8NER1 1/20 0.47
FAAH O00519 1/20 0.44
EPHX2 P34913 1/20 0.44
SCN9A Q15858 1/20 0.44
GCGR P47871 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6685498 0.91 CTSS (0.51) CTSSCTSLCTSKFAAHEPHX2
SCHEMBL6685630 0.90 NPC1 (0.51) CTSSCTSLCTSKTRPV1EPHX2
SCHEMBL6689357 0.89 CTSS (0.50) CTSSCTSLCTSKTRPV1FAAH
SCHEMBL6693346 0.89 CTSS (0.69) CTSSCTSLCTSK
SCHEMBL6690062 0.87 CTSS (0.48) CTSSCTSLCTSKTRPV1EPHX2
SCHEMBL6691227 0.84 CTSS (0.48) CTSSCTSLCTSKEPHX2
SCHEMBL6690343 0.83 CTSS (0.59) CTSSCTSLCTSK
SCHEMBL6686619 0.83 CTSS (0.46) CTSSCTSLCTSK
SCHEMBL6686273 0.83 CTSS (0.46) CTSSCTSLCTSKTRPV1
SCHEMBL5843630 0.82 CTSS (0.81) CTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084842-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed