SCHEMBL6690754

SCHEMBL6690754

O=C(O)c1nc(Br)n(Cc2ccccc2)c1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.51
GAA P10253 2/20 0.51
TSHR P16473 2/20 0.51
CCR2 P41597 1/20 0.44
HPGD P15428 1/20 0.43
RAB9A P51151 2/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
FOLH1 Q04609 1/20 0.42
GPR35 Q9HC97 1/20 0.41
NOTUM Q6P988 1/20 0.41
ALDH1A1 P00352 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
LMNA P02545 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6692683 0.85 ALDH1A1 (0.50) PKMGAATSHRCCR2ALDH1A1
SCHEMBL8861166 0.79 TSHR (0.46) PKMGAATSHRCCR2HPGD
SCHEMBL17140103 0.77 CCR2 (0.43) TSHRCCR2ALDH1A1CYP1A2CYP2D6
SCHEMBL7883606 0.76 POLB (0.46) PKMGAATSHRRAB9ALMNA
SCHEMBL7883305 0.74 TSHR (0.44) PKMGAATSHRCCR2HPGD
SCHEMBL10844803 0.72 KMT2A (0.55) PKMGAATSHRNOTUMALDH1A1
SCHEMBL10844806 0.72 MEN1 (0.51) PKMGAAHPGDALDH1A1SMN1; SMN2
SCHEMBL23421379 0.72 TSHR (0.52) PKMGAATSHRHPGDRAB9A
SCHEMBL8823072 0.71 ALDH1A1 (0.51) PKMGAATSHRCCR2HPGD
SCHEMBL20534213 0.71 LMNA (0.48) TSHRHPGDRAB9AADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004108730-A1 1H-IMIDAZO`4,5-D!PYRIDAZINES AS DPP-IV INHIBITORS FOR THE TREATMENT OF NIDDM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-12-16 WO disclosed