SCHEMBL7883305

SCHEMBL7883305

COC(C)c1nc(C(=O)O)c(C(=O)O)n1Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
CCR2 P41597 2/20 0.38
NOTUM Q6P988 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7887627 0.86 MAPK8 (0.46) GAAPKMSMN1; SMN2KMT2AMAPK8
SCHEMBL8861166 0.84 TSHR (0.46) TSHRGAAPKMCCR2NOTUM
SCHEMBL7883606 0.76 POLB (0.46) TSHRGAAPKMLMNAKMT2A
SCHEMBL6690754 0.74 PKM (0.51) TSHRGAAPKMCCR2NOTUM
SCHEMBL5052843 0.72 TLR7 (0.45) TSHRGAAPKMCCR2NOTUM
SCHEMBL7878415 0.69 TSHR (0.48) TSHRGAALMNASMN1; SMN2HPGD
SCHEMBL15997829 0.66 NOTUM (0.56) TSHRGAAPKMCCR2NOTUM
SCHEMBL8861479 0.66 TLR7 (0.65)
SCHEMBL3363334 0.64 MAPK8 (0.53) TSHRGAAPKMNOTUMSMN1; SMN2
SCHEMBL8823072 0.64 ALDH1A1 (0.51) TSHRGAAPKMCCR2NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573218-B1 4-Carboxyimidazoles as angiotensin II antagonists and their thrapeutic use SANKYO CO (JP) 2001-03-07 EP disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
EP-0573218-A2 4-Carboxyimidazoles as angiotensin II antagonists and their thrapeutic use SANKYO COMPANY LIMITED (JP) 1993-12-08 EP disclosed