Maleic Acid

Maleic Acid

SCHEMBL6691185

C=C(C)OCC.O=C(O)/C=C\C(=O)O

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.61
ALDH1A1 P00352 5/20 0.44
LMNA P02545 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TSHR P16473 3/20 0.41
TP53 P04637 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
EGLN3 Q9H6Z9 1/20 0.41
GLO1 Q04760 1/20 0.39
ALOX15 P16050 1/20 0.37
MGAM O43451 1/20 0.37
GAA P10253 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
SOAT1 P35610 1/20 0.37
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL31496494 0.85 ALDH1A1 (0.52) HCAR2ALDH1A1LMNAHSD17B10TSHR
Maleic Acid SCHEMBL720767 0.83 HCAR2 (0.57) HCAR2ALDH1A1LMNAHSD17B10TSHR
Ethyl Fumarate SCHEMBL27952657 0.83 HCAR2 (0.83) HCAR2ALDH1A1LMNAHSD17B10
Fumaric Acid SCHEMBL8953356 0.83 HCAR2 (0.57) HCAR2ALDH1A1LMNAHSD17B10TSHR
Maleic Acid SCHEMBL15653018 0.83 HCAR2 (0.57) HCAR2ALDH1A1LMNAHSD17B10TSHR
Ethyl Fumarate SCHEMBL8073557 0.82 HCAR2 (0.74) HCAR2ALDH1A1LMNAHSD17B10GLO1
SCHEMBL4899159 0.82 HCAR2 (0.61) HCAR2ALDH1A1LMNAHSD17B10TSHR
SCHEMBL4895205 0.82 HCAR2 (0.61) HCAR2ALDH1A1LMNAHSD17B10TSHR
SCHEMBL17300570 0.82 HCAR2 (0.61) HCAR2ALDH1A1LMNAHSD17B10TSHR
Maleic Acid SCHEMBL6600336 0.81 ALDH1A1 (0.70) HCAR2ALDH1A1LMNAHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040136921-A1 Product containing a clear hair lotion sprayable as an aerosol spray WELLA AKTIENGESELLSCHAFT (DE) 2004-07-15 US disclosed