SCHEMBL6693470

SCHEMBL6693470

CNC(=O)C(NCc1ccc(OCc2c(F)cccc2Cl)cc1OC)C(C)O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
CD274 Q9NZQ7 3/20 0.43
MAOB P27338 2/20 0.41
MAOA P21397 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PDCD1 Q15116 2/20 0.41
CASP1 P29466 2/20 0.40
CASP3 P42574 2/20 0.40
CASP7 P55210 2/20 0.40
CASP8 Q14790 2/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
GAA P10253 1/20 0.40
TP53 P04637 1/20 0.39
PARP15 Q460N3 1/20 0.39
PARP10 Q53GL7 1/20 0.39
STING1 Q86WV6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687664 0.84 MAOB (0.59) LMNACD274MAOBMAOAPARP15
SCHEMBL6687667 0.84 MAOB (0.59) LMNACD274MAOBMAOAPARP15
SCHEMBL6691050 0.83 KMT2A (0.43) LMNACD274MAOBMAOASMN1; SMN2
SCHEMBL6691044 0.83 KMT2A (0.43) LMNACD274MAOBMAOASMN1; SMN2
SCHEMBL6691043 0.81 CD274 (0.51) CD274MAOBPDCD1
SCHEMBL6685871 0.81 CD274 (0.51) CD274MAOBPDCD1
SCHEMBL6685476 0.81 MAOB (0.47) LMNACD274MAOBMAOASMN1; SMN2
SCHEMBL6685482 0.81 MAOB (0.47) LMNACD274MAOBMAOASMN1; SMN2
SCHEMBL6690944 0.78 MAOB (0.48) LMNACD274MAOBMAOATP53
SCHEMBL6685594 0.77 SCN9A (0.50) MAOBMAOAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed