Isonicotinonitrile

Isonicotinonitrile

SCHEMBL669363

N#Cc1ccncc1.O=S(=O)(O)C(F)(F)F

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 4/20 0.48
CYP3A4 P08684 1/20 0.41
CYP3A5 P20815 1/20 0.41
KIF11 P52732 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
CYP19A1 P11511 2/20 0.39
NAMPT P43490 3/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
PTPN5 P54829 1/20 0.37
TRPV4 Q9HBA0 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC8 Q9BY41 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzonitrile SCHEMBL27664681 0.81 TSHR (0.56) SLC22A12KIF11PTPN5TRPV4HDAC1
4-Cyanophenol SCHEMBL28386261 0.79 CA2 (0.61) SLC22A12KIF11CYP19A1CA12CA1
Isonicotinonitrile SCHEMBL1358990 0.79 SLC22A12 (0.43) SLC22A12CYP3A4CYP3A5KIF11CYP19A1
Isonicotinonitrile SCHEMBL2015834 0.77 HDAC8 (0.52) KIF11CYP19A1GAAKMT2ACA12
Isonicotinonitrile SCHEMBL151611 0.77
Isonicotinonitrile SCHEMBL12264099 0.77
Trifluoromethanesulfonic Acid SCHEMBL5069402 0.76 USP2 (0.45) KIF11PTGS1PTGS2NAMPTKMT2A
Trifluoromethanesulfonic Acid SCHEMBL30504299 0.76 KIF11 (0.50) SLC22A12KIF11CYP19A1NAMPTKMT2A
Isonicotinonitrile SCHEMBL27508878 0.75 HDAC8 (0.46) SLC22A12CYP19A1GAAKMT2APOLB
Trifluoromethanesulfonic Acid SCHEMBL2826879 0.75 PTPN5 (0.53) SLC22A12KIF11CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140018538-A1 HIGH-VALENT PALLADIUM FLUORIDE COMPLEXES AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-01-16 US disclosed
EP-2606056-A2 HIGH-VALENT PALLADIUM FLUORIDE COMPLEXES AND USES THEREOF President and Fellows of Harvard College (US) 2013-06-26 EP disclosed
WO-2012024604-A2 HIGH-VALENT PALLADIUM FLUORIDE COMPLEXES AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140018538-A1 HIGH-VALENT PALLADIUM FLUORIDE COMPLEXES AND USES THEREOF NECTIN4, FIS1, DNM1 SLC22A12 1085/4885CYP3A4 2356/4885CYP3A5 3183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.