SCHEMBL6695582

SCHEMBL6695582

NC(=O)c1c[nH]nc1-c1nc2cc(C(F)(F)F)ccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.45
CHEK2 O96017 4/20 0.44
MAP2K4 P45985 1/20 0.42
NPBWR1 P48145 5/20 0.41
FLT3 P36888 1/20 0.41
PDPK1 O15530 1/20 0.40
DGAT1 O75907 3/20 0.39
KCNH2 Q12809 3/20 0.39
SOAT1 P35610 1/20 0.38
CHEK1 O14757 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5951708 0.82 NPBWR1 (0.45) NPBWR1FLT3PDPK1DGAT1KCNH2
SCHEMBL5951733 0.79 CHEK1 (0.39) NPBWR1FLT3PDPK1DGAT1KCNH2
SCHEMBL13374038 0.79 DYRK1A (0.44) NPBWR1FLT3PDPK1DGAT1KCNH2
SCHEMBL5952391 0.78 ALDH1A1 (0.41) NPBWR1FLT3PDPK1DGAT1KCNH2
SCHEMBL5951462 0.78 KIF11 (0.43) NPBWR1PDPK1DGAT1KCNH2SOAT1
SCHEMBL5953146 0.77 HPSE (0.45) CHEK2
SCHEMBL4469806 0.76 PARP1 (0.52) PARP1CHEK2NPBWR1DGAT1KCNH2
SCHEMBL6283906 0.76 CHEK2 (0.40) CHEK2CHEK1
SCHEMBL19994513 0.76 CHEK2 (0.65) PARP1CHEK2MAP2K4NPBWR1DGAT1
SCHEMBL13374039 0.76 PDPK1 (0.46) PDPK1DGAT1KCNH2CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441725-A1 BENZIMIDAZOLES AND ANALOGUES AND THEIR USE AS PROTEIN KINASES INHIBITORS Aventis Pharmaceuticals Inc. (US) 2004-08-04 EP disclosed
WO-2003035065-A1 BENZIMIDAZOLES AND ANALOGUES AND THEIR USE AS PROTEIN KINASES INHIBITORS AVENTIS PHARMACEUTICALS INC (US) 2003-05-01 WO disclosed