SCHEMBL6695838

SCHEMBL6695838

Cc1nc[nH]c1CN1c2ccccc2CC(Cc2ccc(C(C)(C)C)cc2)C(=O)N1CCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.39
ALDH1A1 P00352 3/20 0.35
MAPK1 P28482 1/20 0.35
TSHR P16473 1/20 0.35
SIGMAR1 Q99720 2/20 0.35
TMEM97 Q5BJF2 1/20 0.35
DRD2 P14416 2/20 0.34
DRD4 P21917 1/20 0.34
HDAC6 Q9UBN7 1/20 0.33
GAA P10253 2/20 0.32
KMT2A Q03164 2/20 0.32
MAPT P10636 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
MEN1 O00255 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6694523 0.86 ALDH1A1 (0.35) CYP2C9ALDH1A1MAPK1TSHRSIGMAR1
SCHEMBL6695836 0.85 CYP2C9 (0.37) CYP2C9ALDH1A1TSHRSIGMAR1DRD2
SCHEMBL6694520 0.71 HTT (0.35) CYP2C9ALDH1A1SIGMAR1DRD2DRD4
SCHEMBL6701647 0.71 MAPK1 (0.39) ALDH1A1MAPK1TSHRHDAC6GAA
SCHEMBL6701976 0.71 MTNR1A (0.36) CYP2C9DRD2
SCHEMBL7255593 0.68 HDAC6 (0.34) CYP2C9ALDH1A1TSHRSIGMAR1TMEM97
SCHEMBL30489343 0.65 DRD2 (0.46) ALDH1A1MAPK1TSHRDRD2DRD4
SCHEMBL28995160 0.65 DRD2 (0.46) ALDH1A1MAPK1TSHRDRD2DRD4
SCHEMBL7255157 0.65 MTNR1A (0.36)
SCHEMBL6701125 0.62 CYP2C9 (0.44) CYP2C9ALDH1A1SIGMAR1TMEM97NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040009972-A1 Benzodiazepine inhibitors of mitochondial F1F0 ATP hydrolase and methods of inhibiting F1F0 ATP hydrolase BRISTOL-MYERS COMPANY 2004-01-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009972-A1 Benzodiazepine inhibitors of mitochondial F1F0 ATP hydrolase and methods of inhibiting F1F0 ATP hydrolase MT-ATP6, MT-CO1, ATP5ME CYP2C9 229/4885ALDH1A1 1084/4885MAPK1 4076/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.