SCHEMBL6700869

SCHEMBL6700869

CC(C)(C)c1ccc(CNc2cc(NCc3csc4ccc(Cl)cc34)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 1/20 0.46
CA2 P00918 1/20 0.42
CYP2A6 P11509 3/20 0.41
MAPT P10636 1/20 0.41
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
TRPA1 O75762 1/20 0.37
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PKM P14618 1/20 0.36
CTNNB1 P35222 1/20 0.35
TCF7L2 Q9NQB0 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GAB1 Q13480 1/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6697152 0.89 MAPT (0.47) CA2CYP2A6MAPTKEAP1NFE2L2
SCHEMBL6694360 0.85 P2RX1 (0.47) P2RX1CA2CYP2A6MAPTKEAP1
SCHEMBL6692115 0.82 MEN1 (0.47) P2RX1CA2CYP2A6MAPTSMN1; SMN2
SCHEMBL6696014 0.78 CA1 (0.50) P2RX1CA2TRPV1TRPA1CYP1A2
SCHEMBL6692355 0.77 ADRA2A (0.49) P2RX1CA2TRPV1TRPA1
SCHEMBL6695173 0.72 MAPT (0.51) CA2CYP2A6MAPTKEAP1NFE2L2
SCHEMBL6693244 0.72 MAPT (0.50) CA2CYP2A6MAPTKEAP1NFE2L2
SCHEMBL6691557 0.70 FFAR1 (0.54) P2RX1TRPA1HDAC6
SCHEMBL1241369 0.70 CA1 (0.45) P2RX1CA2TRPV1TRPA1
SCHEMBL17788644 0.70 CA2 (0.58) CA2CYP2A6MAPTKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040009973-A1 Phenylenediamine derivatives N-substituted with benzyl- or heteroarylmethyl- groups 4SC AG (DE) 2004-01-15 US disclosed
WO-2003076388-A2 BIS-ANILINE DERIVATIVES USEFUL AS POTASSIUM CHANNELS MODULATORS 4SC AG (DE) 2003-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009973-A1 Phenylenediamine derivatives N-substituted with benzyl- or heteroarylmethyl- groups PAH, PNMT, OPRM1 P2RX1 1634/4885CA2 1332/4885CYP2A6 68/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.